AKT Kinase Inhibitor

Product Name : AKT Kinase InhibitorDescription:AKT Kinase Inhibitor is an Akt kinase inhibitor with anti-tumor activity.CAS: 842148-40-7Molecular Weight:357.37Formula: C16H19N7O3Chemical Name: 3-[2-(4-amino-1,2,5-oxadiazol-3-yl)-7-(3-aminopropoxy)-1-ethyl-1H-imidazo[4,5-c]pyridin-4-yl]prop-2-yn-1-olSmiles : CCN1C2=C(C=NC(C#CCO)=C2N=C1C1=NON=C1N)OCCCNInChiKey: LWLOLQIXHMFYND-UHFFFAOYSA-NInChi : InChI=1S/C16H19N7O3/c1-2-23-14-11(25-8-4-6-17)9-19-10(5-3-7-24)12(14)20-16(23)13-15(18)22-26-21-13/h9,24H,2,4,6-8,17H2,1H3,(H2,18,22)Purity: ≥98% (or refer to…

Raltegravir (potassium salt)

Product Name : Raltegravir (potassium salt)Description:Raltegravir, also known as MK-0518, is an antiretroviral drug used to treat HIV infection. Raltegravir is a human immunodeficiency virus (HIV) integrase strand transfer inhibitor…

β-glycosidase-IN-1

Product Name : β-glycosidase-IN-1Description:β-glycosidase-IN-1 (Compound 33) is a piperidine derivative and a β-glycosidase inhibitor. β-glycosidase-IN-1 has hypoglycemic activity.CAS: 176485-27-1Molecular Weight:273.33Formula: C13H23NO5Chemical Name: tert-butyl (3aS,7R,7aR)-3a,7a-dihydrogenio-7-hydroxy-2,2-dimethyl-hexahydro-2H-[1,3]dioxolo[4,5-c]pyridine-5-carboxylateSmiles : CC(C)(C)OC(=O)N1C[C@@H]2OC(C)(C)O[C@@H]2[C@H](O)C1InChiKey: RPFDMDWEBWOMNO-KXUCPTDWSA-NInChi : InChI=1S/C13H23NO5/c1-12(2,3)19-11(16)14-6-8(15)10-9(7-14)17-13(4,5)18-10/h8-10,15H,6-7H2,1-5H3/t8-,9+,10-/m1/s1Purity: ≥98%…

Sauristolactam

Product Name : SauristolactamDescription:Sauristolactam, a natural aristolactam isolated from aerial portions of Saururus chinensis, has significant neuroprotective activity against glutamate-induced toxicity in primary cultured rat cortical cells. Sauristolactam also inhibits…

FPH2 (BRD-9424)

Product Name : FPH2 (BRD-9424)Description:FPH2 (BRD-9424) is a small molecule, which promotes differentiation of iPS-derived hepatocytes.CAS: 957485-64-2Molecular Weight:353.83Formula: C14H16ClN5O2SChemical Name: 4-{[(5-chloro-2-methoxyphenyl)carbamothioyl]amino}-1-ethyl-1H-pyrazole-3-carboxamideSmiles : CCN1C=C(NC(=S)NC2C=C(Cl)C=CC=2OC)C(=N1)C(N)=OInChiKey: PCHRYHSDDPPZBV-UHFFFAOYSA-NInChi : InChI=1S/C14H16ClN5O2S/c1-3-20-7-10(12(19-20)13(16)21)18-14(23)17-9-6-8(15)4-5-11(9)22-2/h4-7H,3H2,1-2H3,(H2,16,21)(H2,17,18,23)Purity: ≥98% (or refer to…

3, 3′-Difluorobenzaldazine

Product Name : 3, 3'-DifluorobenzaldazineDescription:3,3'-Difluorobenzaldazine (DFB) is a selective positive allosteric modulator of mGluR5. 3,3'-Difluorobenzaldazine potentiates 3- to 6-fold action for mGlu5 agonists (Glutamate, Quisqualate, and 3,5-Dihydroxyphenylglycine), with EC50s in…

GNE-207

Product Name : GNE-207Description:GNE-207 is a potent, selective and orally bioavailable inhibitor of the bromodomain of CBP, with an IC50 of 1 nM, exhibits a selectively index of >2500-fold against BRD4…

Tazemetostat trihydrochloride

Product Name : Tazemetostat trihydrochlorideDescription:Tazemetostat trihydrochloride (EPZ-6438 trihydrochloride) is a potent, selective and orally available EZH2 inhibitor. Tazemetostat trihydrochloride inhibits the activity of human polycomb repressive complex 2 (PRC2)-containing wild-type…